Beyond Peptides and Peptidomimetics: Natural Heteroaromatic Amino Acids in the Synthesis of Fused Heterocyclic Frameworks for Bioactive Agents
Isis Apolo Silveira de Borba, Jamile Buligon Peripolli, Angélica Rocha Joaquim & Fernando Fumagalli · Organics · 2025
Heterocycle cores are widely used in medicinal chemistry for developing bioactive compounds. In this scenario, using cheap and accessible starting material to build these heterocycles is desirable to obtain new drug candidates for cost-efficient processes. One easily accessible s...
Open access
Research Article
10.3390/org6020023